A practical route to quinolines from anilines

Hidetoshi Tokuyama; Masashi Sato; Toshihiro Ueda; Tohru Fukuyama

doi:10.3987/com-00-s(i)63

A practical route to quinolines from anilines

Hidetoshi Tokuyama, Masashi Sato, Toshihiro Ueda, Tohru Fukuyama

PHA - Molecular Pharmaceutical Science

The University of Tokyo

Research output: Contribution to journal › Article › peer-review

41 Citations (Scopus)

Abstract

A practical route to quinoline from anilines through acid-mediated cyclization of 3-(N-aryl-N-sulfonylamino)propionaldehydes has been developed. Treatment of the cyclization products, dihydroquinoline intermediates with KOH in DMSO leads to substituted quinolines.

Original language	English
Pages (from-to)	105-108
Number of pages	4
Journal	Heterocycles
Volume	54
Issue number	1
DOIs	https://doi.org/10.3987/com-00-s(i)63
Publication status	Published - 2001 Jan 1

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AU - Ueda, Toshihiro

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A practical route to quinolines from anilines

Abstract

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