Synthesis of eudistomin C and E: Improved preparation of the indole unit

Hiroaki Yamagishi; Koji Matsumoto; Kotaro Iwasaki; Tohru Miyazaki; Satoshi Yokoshima; Hidetoshi Tokuyama; Tohru Fukuyama

doi:10.1021/ol800527p

Synthesis of eudistomin C and E: Improved preparation of the indole unit

Hiroaki Yamagishi, Koji Matsumoto, Kotaro Iwasaki, Tohru Miyazaki, Satoshi Yokoshima, Hidetoshi Tokuyama, Tohru Fukuyama

PHA - Molecular Pharmaceutical Science

The University of Tokyo

Research output: Contribution to journal › Article › peer-review

19 Citations (Scopus)

Abstract

(Chemical Equation Presented) An improved synthesis of the indole unit, a key intermediate for eudistomin C, was established utilizing Makosza's indole synthesis. A concise total synthesis of eudistomin E was achieved on the basis of the improved synthesis.

Original language	English
Pages (from-to)	2369-2372
Number of pages	4
Journal	Organic Letters
Volume	10
Issue number	12
DOIs	https://doi.org/10.1021/ol800527p
Publication status	Published - 2008

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10.1021/ol800527p

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title = "Synthesis of eudistomin C and E: Improved preparation of the indole unit",

abstract = "(Chemical Equation Presented) An improved synthesis of the indole unit, a key intermediate for eudistomin C, was established utilizing Makosza's indole synthesis. A concise total synthesis of eudistomin E was achieved on the basis of the improved synthesis.",

author = "Hiroaki Yamagishi and Koji Matsumoto and Kotaro Iwasaki and Tohru Miyazaki and Satoshi Yokoshima and Hidetoshi Tokuyama and Tohru Fukuyama",

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doi = "10.1021/ol800527p",

language = "English",

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journal = "Organic Letters",

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TY - JOUR

T1 - Synthesis of eudistomin C and E

T2 - Improved preparation of the indole unit

AU - Yamagishi, Hiroaki

AU - Matsumoto, Koji

AU - Iwasaki, Kotaro

AU - Miyazaki, Tohru

AU - Yokoshima, Satoshi

AU - Tokuyama, Hidetoshi

AU - Fukuyama, Tohru

PY - 2008

Y1 - 2008

N2 - (Chemical Equation Presented) An improved synthesis of the indole unit, a key intermediate for eudistomin C, was established utilizing Makosza's indole synthesis. A concise total synthesis of eudistomin E was achieved on the basis of the improved synthesis.

AB - (Chemical Equation Presented) An improved synthesis of the indole unit, a key intermediate for eudistomin C, was established utilizing Makosza's indole synthesis. A concise total synthesis of eudistomin E was achieved on the basis of the improved synthesis.

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U2 - 10.1021/ol800527p

DO - 10.1021/ol800527p

M3 - Article

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AN - SCOPUS:48849112883

SN - 1523-7060

VL - 10

SP - 2369

EP - 2372

JO - Organic Letters

JF - Organic Letters

IS - 12

ER -

Synthesis of eudistomin C and E: Improved preparation of the indole unit

Abstract

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